Substituted cyclohexylaminopyrimidines

US6197729A · kind A · utility

Assignee

• Hoechst Schering Agrevo GmbH · DE

Inventors

• Martin Markl · Frankfurt, DE
• Wolfgang Schaper · Diedorf, DE
• Oswald Ort · Königstein, DE
• Harald Jakobi · Frankfurt, DE
• Ralf Braun · Ramberg, DE
• Gerhard Krautstrunk · Bad Vilbel, DE
• Ulrich Sanft · Hofheim, DE
• Werner Bonin · Kelkheim, DE
• Herbert Stark · Kelkheim, DE
• Sergej Pasenok · Kelkheim, DE
• Ivan Cabrera · Dreieich, DE

Key dates

• Filing date: Jul 29, 1999
• Grant date: Mar 6, 2001
• Expiry date: Jul 29, 2019

Classification

• Technology area (CPC C): Chemistry; Metallurgy
• CPC primary: C07D239/47
• WIPO field: Organic fine chemistry
• WIPO sector: Chemistry

Abstract

Compounds of formula I ##STR1## where PA1 R.sup.1 is hydrogen, chlorine, fluorine or methyl, PA1 R.sup.2 and R.sup.3, which may be the same or different from each other, are hydrogen, halogen, cyano, (C.sub.1 -C.sub.4)-alkyl, vinyl, ethynyl, (C.sub.1 -C.sub.4)-alkoxy, (C.sub.1 -C.sub.4)-alkoxy-(C.sub.1 -C.sub.4)-alkyl, fluorovinyl or fluoroethyl, or PA1 R.sup.2 and R.sup.3 together with the linking carbon atoms form a benzo ring, and PA1 R.sup.4 is (C.sub.2 -C.sub.4)-alkyl, (C.sub.2 -C.sub.4)-alkenyl or (C.sub.3 -C.sub.4)-alkinyl, each of which is substituted by at least two fluorine atoms and optionally substituted by C.sub.1-4 -alkoxy, cyanomethoxy, (C.sub.3 -C.sub.4)-alkenyloxy or (C.sub.3 -C.sub.4)-alkinyloxy, are useful as pesticides, especially against insects, acarids and fungi. The invention includes a novel process for fluorinating certain pyrimidines.