Patent · US Expired

Synthesis of epothilones, intermediates thereto and analogues thereof

US6204388A · kind A · utility

73Cited by
3References
9Claims
0Family size

Assignee

Inventors

Key dates

Filing dateFeb 24, 1999
Grant dateMar 20, 2001
Priority date
Expiry dateFeb 24, 2019

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07F7/1892
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides convergent processes for preparing epothilone A and B, desoxyepothilones A and B, and analogues thereof, useful in the treatment of cancer and cancer which has developed a multidrug-resistant phenotype. Also provided are intermediates useful for preparing said epothilones.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.