Patent · US Expired

Tricyclic amide and urea compounds useful for inhibition of G-protein function and for treatment of proliferative diseases

US6242458A · kind A · utility

9Cited by
13References
8Claims
0Family size

Assignee

Inventors

Key dates

Filing dateSep 21, 1999
Grant dateJun 5, 2001
Priority date
Expiry dateSep 21, 2019

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D417/14
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A method of inhibiting Ras function and therefore inhibiting the abnormal growth of cells is disclosed. The method comprises the administration of a compound of Formula 1.0: ##STR1## to a biological system. In particular, the method inhibits the abnormal growth of cells in a mammal such as a human being. Novel compounds of the formulas 5.1 and 5.2 are disclosed. ##STR2## ##STR3##

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.