Patent · US Expired

Aminotriazole compounds

US6245916A · kind A · utility

16Cited by
0References
13Claims
0Family size

Assignee

Inventors

Key dates

Filing dateApr 14, 2000
Grant dateJun 12, 2001
Priority date
Expiry dateApr 14, 2020

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02P20/55
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compound of formula (I): ##STR1## wherein: PA1 n is 0 or 1, PA1 W represents --CO-- or S(O).sub.q and q is 0, 1 or 2, PA1 G represents a G.sub.1, G.sub.2, G.sub.3 or G.sub.4 group as defined in the description, PA1 Z represents alkyl, aryl, heteroaryl, arylalkyl, arylalkenyl, arylalkynyl, heteroarylalkenyl, heteroarylalkynyl or heteroarylalkyl each optionally substituted. PA1 A represents a grouping selected from --A.sub.2 --, --A.sub.1 --A.sub.2 --, --A.sub.2 --A.sub.1 -- and --A.sub.1 --A.sub.2 --A.sub.1 -- wherein A.sub.1 is alkylene and A.sub.2 represents phenylene, cycloalkylene, naphthylene or heteroarylene each optionally substituted, PA1 R represents hydrogen, alkyl, aryl, heteroaryl, arylalkyl arylalkenyl, arylalkynyl, heteroarylakenyl, heteroarylalkynyl or heteroarylalkenyl each optionally substituted, PA1 R.sub.1 represents alkyl, aryl, heteroary, arylalkyl arylalkenyl, arylalkynyl, heteroarylalkenyl, heteroarylalkynyl or heteroarylalkyl each optionally substituted, and medicinal products containing the same which are useful as Neuropeptide Y receptor ligands.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.