Patent · US Expired

Extended release acetaminophen

US6254891A · kind A · utility

5Cited by
7References
2Claims
0Family size

Assignee

Inventors

Key dates

Filing dateSep 3, 1998
Grant dateJul 3, 2001
Priority date
Expiry dateSep 3, 2018

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K9/5078
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

An extended release acetaminophen composition comprises particles containing acetaminophen coated on sugar/starch seeds. The particles are present as a blend of both an immediate release and a controlled release form. The composition, when contained within a gelatin capsule and assayed in a USP Apparatus I rotating basket at 50 rpm in 900 mL of phosphate buffer at pH 5.8 and a temperature of 37.degree. C., exhibits about 40 percent acetaminophen dissolution at one-half hour, about 55 percent acetaminophen dissolution at one hour, and substantially complete dissolution of acetaminophen at six hours. A process for treating a human patient with the extended release acetaminophen composition is also disclosed.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.