Patent · US Expired

Azetidinylpropylpiperidine derivatives, intermediates and use as tachykinin antagonists

US6262046A · kind A · utility

13Cited by
2References
22Claims
0Family size

Assignee

Inventors

Key dates

Filing dateNov 10, 1999
Grant dateJul 17, 2001
Priority date
Expiry dateNov 10, 2019

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D403/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compounds of the formula (I): ##STR1## where X.sup.1, A, Ar.sup.1, X and R are as defined in the specification, and pharmaceutically-acceptable salts thereof, are new, and are useful as tachykinin inhibitors which act at the NK.sub.1, NK.sub.2 and NK.sub.3 receptors or a combination of two or more thereof.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.