Cycloalkano-indole and -azaindole derivatives

US6265431A · kind A · utility

Assignee

• BAYER HEALTHCARE LLC · DE

Inventors

• Ulrich Muller · Wuppertal, DE
• Richard Connell · Trumbull, US
• Siegfried Goldmann · Wuppertal, DE
• Rudi Grutzmann · Solingen, DE
• Martin Beuck · Milford, US
• Hilmar Bischoff · Wuppertal, DE
• Dirk Denzer · Wuppertal, DE
• Anke Domdey-Bette · Hückeswagen, DE
• Stefan Wohlfeil · Hilden, DE

Key dates

• Filing date: May 17, 1999
• Grant date: Jul 24, 2001
• Expiry date: May 17, 2019

Classification

• Technology area (CPC C): Chemistry; Metallurgy
• CPC primary: C07D219/02
• WIPO field: Pharmaceuticals
• WIPO sector: Chemistry

Abstract

Cycloalkano-indole and -azaindole derivatives are prepared by reaction of appropriately substituted carboxylic acids with amines. The cycloalkano-indole and -azaindole derivatives are suitable as active compounds for medicaments, preferably antiatherosclerotic medicaments.