Patent · US Expired

Fenofibrate pharmaceutical composition having high bioavailability and method for preparing it

US6277405A · kind A · utility

33Cited by
6References
13Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 18, 2000
Grant dateAug 21, 2001
Priority date
Expiry dateMay 18, 2020

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K9/2081
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention provides a micronized fenofibrate composition. The micronized fenofibrate composition has a dissolution of at least 10% in 5 minutes, 20% in 10 minutes, 50% in 20 minutes and 75% in 30 minutes, as measured using the rotating blade method at 75 rpm according to the European Pharmacopoeia, in a dissolution medium constituted by water with 2% by weight polysorbate 80 or with 0.025M sodium lauryl sulfate. The composition can further comprise hydrophilic polymers, surfactants, hydrosoluble carriers, outer phases or layers, or other pharmaceutically acceptable excipients. The immediate-release fenofibrate composition is preferably in the form of a tablet or in the form of granules inside a capsule.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.