Patent · US Expired

Chemical compounds

US6277880A · kind A · utility

0Cited by
4References
15Claims
0Family size

Assignees

Inventors

Key dates

Filing dateMay 19, 1999
Grant dateAug 21, 2001
Priority date
Expiry dateMay 19, 2019

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07C311/51
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Prodrugs, of generic formula I, are disclosed for use in antibody directed enzyme prodrug therapy (ADEPT). The prodrugs are substrates for carboxypeptidase G2 (CPG2) and yield more active cytotoxic drugs than known products of CPG2 catalysed reactions.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.