Antithrombotic agents

US6284756A · kind A · utility

Assignee

• ELI LILLY AND COMPANY · US

Inventors

• Nickolay Y Chirgadze · Carmel, US
• Richard Waltz Harper · Indianapolis, US
• Todd Johnathan Kohn · Fishers, US
• Ho-Shen Lin · Indianapolis, US
• Jefferson Ray McCowan · Indianapolis, US
• Alan David Palkowitz · Carmel, US
• Daniel Jon Sall · Greenwood, US
• Gerald Floyd Smith · Indianapolis, US
• Kumiko Takeuchi · Indianapolis, US
• Michael Robert Wiley · Zionsville, US
• Minsheng Zhang · Hackettstown, US

Key dates

• Filing date: Jan 21, 2000
• Grant date: Sep 4, 2001
• Expiry date: Jan 21, 2020

Classification

• Technology area (CPC C): Chemistry; Metallurgy
• CPC primary: C07D409/12
• WIPO field: Organic fine chemistry
• WIPO sector: Chemistry

Abstract

This application relates to novel compounds of formula I (and their pharmaceutically acceptable salts), as defined herein, processes and intermediates for their preparation, pharmaceutical formulations comprising the novel compounds of formula I, and the use of the compounds of formula I as thrombin inhibitors.