Patent · US Expired

Acronycine derivatives, preparation method and pharmaceutical compositions

US6288073A · kind A · utility

2Cited by
1References
12Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 19, 2000
Grant dateSep 11, 2001
Priority date
Expiry dateJun 19, 2020

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D491/14
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

A compound selected from those of formula (I): ##STR1## in which: PA1 X and Y represent hydrogen, halogen, hydroxy, mercapto, cyano, nitro, alkyl, alkoxy, trihaloalkyl, optionally substituted amino, methylenedioxy, or ethylenedioxy, PA1 R.sub.1 represents hydrogen, or alkyl, PA1 R.sub.2 represents hydrogen, hydroxy, alkyl, alkoxy, alkylcarbonyloxy, or optionally substituted ammo, PA1 R.sub.3 and R.sub.4 represent hydrogen, or alkyl, PA1 A represents --CH.dbd.CH--, or --CH(R.sub.5)--CH(R.sub.6)-- wherein R.sub.5 and R.sub.6 are as defined in the description, their isomers, N-oxides, and pharmaceutically-acceptable acid or base addition salts thereof, and medicinal products containing the same which are useful in the treatment of cancer.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.