Patent · US Expired

2,3-methano-amino acid compounds

US6288077A · kind A · utility

4Cited by
3References
15Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 2, 2000
Grant dateSep 11, 2001
Priority date
Expiry dateMay 2, 2020

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02P20/55
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compound of formula (I): ##STR1## wherein: PA1 n represents 2 or 3, PA1 R.sub.1 represents optionally substituted alkyl, cycloalkyl or optionally substituted phenyl, PA1 R.sub.2 represents amino, optionally substituted amidino, optionally substituted guanidino or optionally substituted isothioureido, PA1 Ar represents aryl or heteroaryl, PA1 X.sub.1 represents hydroxy or optionally substituted amino, PA1 isomers thereof, and also salts thereof with a pharmaceutically acceptable acid or base, and which PA1 medicinal products containing the same/are useful as trypsin-related serine protease inhibitors.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.