Patent · US Expired

Methods of o-demethylation and n-deprotection

US6291675A · kind A · utility

36Cited by
0References
18Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 6, 1999
Grant dateSep 18, 2001
Priority date
Expiry dateJul 6, 2019

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D489/12
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention provides a method for N-deprotecting an opioid compound, a method for N-deprotecting and O-demethylating an opioid compound, a method for O-demethylating an opioid compound, and a method for O-demethylating a nonpeptidic delta agonist compound or an opioid compound having a tertiary amide with no significant reaction at amide groups.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.