Patent · US Expired

4-[aryl(8-azabicyclo[3.2.1]octan-3-yl)]aminobenzoic acid derivatives

US6306876A · kind A · utility

3Cited by
0References
30Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 4, 2000
Grant dateOct 23, 2001
Priority date
Expiry dateDec 4, 2020

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P43/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

4-[aryl(8-azabicyclo[3.2.1]octan-3yl)]aminobenzoic acid derivatives are delta-opioid receptor modulators. As delta-opioid receptor agonists, such compounds are useful as analgesics. Depending on their antagonist effect, such compounds may also be useful immunosuppressants, antiinflammatory agents, agents for the treatment of neurological and psychiatric conditions, medicaments for drug and alcohol abuse, agents for treating gastritis and diarrhea, cardiovascular agents and agents for the treatment of respiratory diseases.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.