Benzoheterocyclic derivatives
US6335327B1 · kind B1 · utility
6Cited by
16References
20Claims
0Family size
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Inventors
Key dates
| Filing date | Nov 1, 1999 |
| Grant date | Jan 1, 2002 |
| Priority date | — |
| Expiry date | Nov 1, 2019 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D471/04
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
A benzoheterocyclic derivative of the following formula [1]: and pharmaceutically acceptable salts thereof, which show excellent anti-vasopressin activity, vasopressin agonistic activity and oxytocin antagonistic activity, and are useful as a vasopressin antagonist, vasopressin agonist or oxytocin antagonist.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.