Steroid sulfamates, method for the production and use thereof

US6339079B1 · kind B1 · utility

Assignee

• ID Pharma Co., Ltd. · DE

Inventors

• Helmut Kasch · Jena, DE
• Winfried Schumann · Jena, DE
• Johannes Roemer · Großerkmannsdorf, DE
• Joerg Steinbach · Dresden, DE

Key dates

• Filing date: Feb 2, 2000
• Grant date: Jan 15, 2002
• Expiry date: Feb 2, 2020

Classification

• Technology area (CPC Y): Emerging Cross-Sectional Technologies
• CPC primary: Y02P20/55
• WIPO field: Pharmaceuticals
• WIPO sector: Chemistry

Abstract

A novel class of gonane type and D-homo-gonane type steroids having sulfatase-inhibiting and/or estrogenic activity is presented for application in the pharmaceutical industry. The number and location of sulfamoyloxy groups on the steroids provides for sulfatase inhibiting and estrogenic activities that independently vary over a wide range, allowing the customization of the pharmaceutical for specific purposes, including treatment and diagnosis of estrogen-dependent tumors.