Patent · US Expired

Alkynyl containing hydroxamic acid compounds as matrix metalloproteinase and tace inhibitors

US6340691B1 · kind B1 · utility

17Cited by
18References
5Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJan 27, 2000
Grant dateJan 22, 2002
Priority date
Expiry dateJan 27, 2020

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07C2601/14
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Compounds of the formula are useful in treating disease conditions mediated by TNF-&agr;, such as rheumatoid arthritis, osteoarthritis, sepsis, AIDS, ulcerative colitis, multiple sclerosis, Crohn's disease and degenerative cartilage loss.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.