Erythromycin a derivatives and method for preparing same
US6342590B1 · kind B1 · utility
Assignee
Inventors
Key dates
| Filing date | Apr 14, 1992 |
| Grant date | Jan 29, 2002 |
| Priority date | — |
| Expiry date | Apr 14, 2012 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07H17/08
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
Erythromycin A derivatives represented by the general formula wherein R1 is a 2-alkenyl group having 3 to 15 carbon atoms, an arylmethyl group, or an arylmethyl group substituted by 1 to 3 of a halogen atom, an alkoxy group 1 to 4 carbon atoms, a nitro group or an alkoxycarbonyl group having 2 to 6 carbon atoms, R2 is a substituted silyl group and R3 is a hydrogen atom or R2, are disclosed. These compounds are useful as intermediates of the anti-bacterial agents.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.