Solid phase synthesis of heterocycles
US6362009B1 · kind B1 · utility
8Cited by
47References
24Claims
0Family size
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Key dates
| Filing date | Nov 21, 1997 |
| Grant date | Mar 26, 2002 |
| Priority date | — |
| Expiry date | Nov 21, 2017 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D211/86
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
Methods for solid phase and combinatorial synthesis using a resin activation/capture approach are provided. In particular, methods for the production of dihydropyridones, N-acyidihydropyridones, tetrahydropyridones, pyridines, aminopyridines, N-acyltetrahydropyridines and tetrahydropyridines compounds and libraries containing such compounds are provided. Methods for screening the libraries and compounds and pharmaceutical compositions containing compounds prepared by the methods are provided.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.