Patent · US Expired

Farnesyl protein transferase inhibitors

US6362188B1 · kind B1 · utility

22Cited by
4References
29Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 16, 1999
Grant dateMar 26, 2002
Priority date
Expiry dateDec 16, 2019

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D401/14
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Disclosed are compounds of the formula: wherein R8 represents a cyclic moiety to which is bound an imodazolylalkyl group; R9 represents a carbamate, urea, amide or sulfonamide group; and the remaining substituents are as defined herein. Also disclosed is a method of treating cancer and a method of inhibiting farnesyl protein transferase using the disclosed compounds.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.