Patent · US Expired

Quinoline and quinazoline compounds useful in therapy

US6365599B1 · kind B1 · utility

0Cited by
3References
8Claims
0Family size

Assignee

Inventor

Key dates

Filing dateJun 2, 2000
Grant dateApr 2, 2002
Priority date
Expiry dateJun 2, 2020

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D471/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Compounds of formula I, whereinR1 represents C1-4 alkoxy optionally substituted by one or more fluorine atoms;R2 represents H or C1-6 alkoxy optionally substituted by one or more fluorine atoms;R3 represents a 5- or 6-membered heterocyclic ring, the ring being optionally substituted;R4 represents a 4-, 5-, 6-, or 7-membered heterocyclic ring, the ring being optionally fused to a benzene ring or 5- or 6-membered heterocyclic ring, the ring system as a whole being optionally substituted;L is absent;and pharmaceutically acceptable salts thereof; are useful in therapy, in particular in the treatment of benign prostatic hyperplasia.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.