Patent · US Expired

Treatment of mastitis

US6369049B1 · kind B1 · utility

0Cited by
8References
21Claims
0Family size

Assignee

Inventor

Key dates

Filing dateApr 12, 1999
Grant dateApr 9, 2002
Priority date
Expiry dateApr 12, 2019

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D463/20
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention provides new fluorinated cephalosporin antibiotics of Formula I whereinRa, Rb, Rc, Rd and Re, independently, are H, F or a C1-C6 alkyl-(Z)n— group having at least one fluorine substituent;X is O or S;Y is S, O, or —CH2—;Z is O, S, —SO—, or —SO2—;m and n independently are 0 or 1; andR1 is H, C1-C6-alkyl, phenyl or benzyl, each of which may optionally have up to three substituents selected from halo, C1-C4-alkoxy, phenyl, NO2, C1-C6-alkanoyl, benzoyl, or C1-C6-alkanoyloxy; or a physiologically acceptable salt thereof;and methods of preventing or treating or treating infection, particularly mastitis in ruminants, using these antibiotics.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.