Patent · US Expired

Chemical transformation of substrates using nonmetallic, organic catalyst compositions

US6369243B1 · kind B1 · utility

10Cited by
4References
74Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJan 18, 2000
Grant dateApr 9, 2002
Priority date
Expiry dateJan 18, 2020

Classification

  • Technology area (CPC B)Performing Operations; Transporting
  • CPC primaryB01J2231/72
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

A method is provided for catalytically transforming a functional group within a first reactant by reaction with a second reactant in the presence of a nonmetallic, organic catalyst composition composed of a heteroatom-containing activator and an acid, or a salt of a heteroatom-containing activator and an acid. Exemplary first reactants are &agr;,&bgr;-unsaturated carbonyl compounds such as &agr;,&bgr;-unsaturated ketones and &agr;,&bgr;-unsaturated aldehydes. The heteroatom of the activator is a Group 15 or Group 16 element such as nitrogen, oxygen, sulfur or phosphorus, and exemplary heteroatom-containing activators are amines. Chiral heteroatom-containing activators can be used to catalyze enantioselective reactions, such that a chiral product is obtained from a chiral or achiral starting material in enantiomerically pure form.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.