Patent · US Expired

2-decarboxy-2-phosphinico Prostaglandin F analogs

US6372730B1 · kind B1 · utility

13Cited by
5References
14Claims
0Family size

Assignee

Inventors

Key dates

Filing dateAug 3, 2000
Grant dateApr 16, 2002
Priority date
Expiry dateAug 3, 2020

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P27/06
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention provides novel Prostaglandin F analogs. In particular, the present invention is directed to compounds having a structure according to the following formula: wherein R1, R2, X, Y, V, a, b, W, and Z are defined below.This invention also includes optical isomers, diastereomers and enantiomers of the formula above, and pharmaceutically—acceptable salts, biohydrolyzable amides, esters, and imides thereof.The compounds of the present invention are useful for the treatment of a variety of diseases and conditions, such as bone disorders and glaucoma. Accordingly, the invention further provides pharmaceutical compositions comprising these compounds. The invention still further provides methods of treatment for bone disorders and glaucoma using these compounds or the compositions containing them.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.