Patent · US Expired

Process for the manufacture of pharmaceutical composition with modified release of active principle comprising the matrix

US6375987B1 · kind B1 · utility

76Cited by
2References
4Claims
0Family size

Assignee

Inventors

Key dates

Filing dateNov 22, 2000
Grant dateApr 23, 2002
Priority date
Expiry dateNov 22, 2020

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K9/1617
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention relates to a process for the manufacture of a pharmaceutical composition with modified release of active principle comprising at least one active principle, a lipid matrix agent composed of ester of alcohol with at least one fatty acid and at least one adjuvant.This process is characterized in that:a powder composed of at least one component selected in the group comprising the active principle and the adjuvant, is mixed, while heating and fluidizing, in order to obtain individual grains;the said lipid matrix agent is liquefied separately under warm conditions;the said powder is then coated under warm conditions by spraying the said lipid matrix agent over the individual grains;finally, the temperature of the combined product is lowered in order to allow the lipid matrix agent to solidify.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.