Patent · US Expired

Peptide-enhanced transfections

US6376248B1 · kind B1 · utility

142Cited by
32References
30Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 16, 1998
Grant dateApr 23, 2002
Priority date
Expiry dateMar 16, 2018

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC12N2740/16322
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides compositions useful for transfecting eukaryotic cells comprising nucleic acid complexes with peptides, wherein the peptide is optionally covalently coupled to a nucleic acid-binding group, and cationic lipids or dendrimers as transfection agents. The invention also provides transfection compositions in which a peptide is covalently linked to the transfection agent (lipid, cationic lipid or dendrimer). Inclusion of peptides or modified-peptides in transfection compositions or covalent attachment of peptides to transfection agents results in enhanced transfection efficiency. Methods for the preparation of transfection compositions and methods of using these transfection compositions as intracellular delivery agents and extracellular targeting agents are also disclosed.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.