Patent · US Expired

Antifungal azole derivatives having a fluorinated vinyl group and process for preparing same

US6376497B1 · kind B1 · utility

0Cited by
3References
5Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 6, 2001
Grant dateApr 23, 2002
Priority date
Expiry dateJul 6, 2021

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D405/06
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

An antifungal compound of formula (I) or a pharmaceutically acceptable salt thereof: wherein:X is CH or N;Y is O, R1 and R2 are each independently F or Cl;R3 is a thiophenyl, naphthyl, or phenyl group, the phenyl group being optionally substituted with one or more substituents selected from the group consisting of C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy, methylenedioxy and halogen; andR4 is H or trifluoromethyl.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.