Patent · US Expired

Carboxamidothiazole derivatives, preparation, pharmaceutical compositions containing them

US6380230B1 · kind B1 · utility

14Cited by
5References
33Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 2, 2000
Grant dateApr 30, 2002
Priority date
Expiry dateJun 2, 2020

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D417/14
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to cholecystokinin (CCK)-agonist substituted thiazoles of formula: in which R1 is a substituted phenyl group, R2 is a group chosen from CH2—R7, (CH2)2—R7, S—CH2—R7, CH2—S—R7 and (C5-C8)alkyl with R7 being a (C5-C7)cycloalkyl group, and R3 is a group with R8 being a group (CH2)nR15 or and R15 being COOH or COO(C1-C4)alkyl. The invention also relates to a process for the preparation of the pharmaceutical compositions containing them and to their uses for the preparation of medicines.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.