Patent · US Expired

HIV integrase inhibitors

US6380249B1 · kind B1 · utility

22Cited by
9References
21Claims
0Family size

Assignees

Inventors

Key dates

Filing dateJun 1, 1999
Grant dateApr 30, 2002
Priority date
Expiry dateJun 2, 2019

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07C2602/10
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Certain six-membered aromatic and heteroaromatic-dioxobutyric acid derivatives are described as inhibitors of HIV integrase and inhibitors of HIV replication. These compounds are useful in the prevention or treatment of infection by HIV and the treatment of AIDS, either as compounds, pharmaceutically acceptable salts, pharmaceutical composition ingredients, whether or not in combination with other antivirals, immunomodulators, antibiotics or vaccines. Methods of treating AIDS and methods of preventing or treating infection by HIV are also described.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.