Patent · US Expired

4,5,6 and 7-indole and indoline derivatitives, their preparation and use

US6391882B1 · kind B1 · utility

7Cited by
1References
14Claims
0Family size

Assignee

Inventors

Key dates

Filing dateFeb 2, 2001
Grant dateMay 21, 2002
Priority date
Expiry dateFeb 2, 2021

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D413/14
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

A substituted 4-, 5-, 6-, and 7-indole derivative of Formula (I) wherein A is a group having formula (IIA), (IIB), (IIC) wherein X, U, Y, R3 to R12, Z, W, n and m are as defined above. The compounds are potent serotonin reuptake inhibitors and have 5-HT1A receptor antagonistic activity.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.