Patent · US Expired

Kappa agonist compounds and pharmaceutical formulations thereof

US6391910B1 · kind B1 · utility

3Cited by
1References
5Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJan 6, 2000
Grant dateMay 21, 2002
Priority date
Expiry dateJan 6, 2020

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D295/073
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compounds having kappa opioid agonist activity, compositions containing them and method of using them as analgesics are provided.The compounds of formulae I, II, IIA, III, IIIA, IV and IVA have the structure: whereinR1, R2, R3, R4; andX, X4, X5, X7, X9;Y, Z and n are as described in the specification.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.