Substituted thiazol(in) ylideneamino sulfonylamino (thio)carbonyl-triazolinones

US6403535B1 · kind B1 · utility

Assignee

• BAYER HEALTHCARE LLC · DE

Inventors

• Klaus-Helmut Muller · Düsseldorf, DE
• Klaus Konig · Leverkusen, DE
• Johannes-Rudolf Jansen · Monheim, DE
• Ernst Rudolf F. Gesing · Erkrath, DE
• Mark Wilhelm Drewes · Langenfeld, DE
• Markus Dollinger · Leverkusen, DE
• Ingo Wetcholowsky · Mangaratiba, BR

Key dates

• Filing date: Apr 27, 2001
• Grant date: Jun 11, 2002
• Expiry date: Apr 27, 2021

Classification

• Technology area (CPC A): Human Necessities
• CPC primary: A01N47/38
• WIPO field: Organic fine chemistry
• WIPO sector: Chemistry

Abstract

The invention relates to novel substituted thiazol(in)ylidenaminosulphonyl-amino(thio)carbonyl-triazolinones of the formula (I) in whichQ represents oxygen or sulphur,R1 represents hydrogen, amino, alkylideneamino or represents an in each case optionally substituted radical from the group consisting of alkyl, alkoxy, alkylamino, dialkylamino, alkanoylamino, alkenyl, alkinyl, alkenyloxy, cycloalkyl, cycloalkylalkyl, cycloalkylamino, aryl and arylalkyl,R2 represents hydrogen, cyano, halogen or represents an in each case optionally substituted radical from the group consisting of alkyl, alkoxy, alkylthio, alkylsulphinyl, alkylsulphonyl, alkylamino, dialkylamino, alkenyl, alkinyl, alkenyloxy, alkenylthio, alkenylamino, cycloalkyl, cycloalkylalkyl, cycloalkyloxy, cycloalkylthio, cycloalkylamino, aryl, aryloxy, arylthio, arylamino, arylalkyl, arylalkoxy, arylalkylthio and arylalkylamino,R3 represents an in each case optionally substituted radical from the group consisting of alkyl, alkoxy, alkenyl, alkinyl, cycloalkyl, cycloalkylalkyl, aryl and arylalkyl,R4 represents hydrogen, cyano, halogen or optionally substituted alkyl,R5 represents hydrogen, cyano, halogen or optionally substituted…