Patent · US Expired

Synthesis of carbamate ketolide antibiotics

US6403776B1 · kind B1 · utility

0Cited by
3References
66Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 5, 2000
Grant dateJun 11, 2002
Priority date
Expiry dateJul 27, 2020

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07H17/08
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The invention relates to a method of preparing a macrolide antibiotic of the formula wherein R1, R2, R3, R4, R5 are defined above. These antibiotics are useful as antibacterial and antiprotozoal agents in mammals, including man, as well as in fish and birds. The invention also includes novel compounds made by the preparation of the macrolide antibiotic.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.