Patent · US Expired

Naphthylsalicylanilides as antimicrobial and antiinflammatory agents

US6407288B1 · kind B1 · utility

2Cited by
5References
27Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 2, 2001
Grant dateJun 18, 2002
Priority date
Expiry dateOct 2, 2021

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07C235/84
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention discloses novel naphthylsalicylanilides of the general formula wherein W is a substituted or unsubstituted naphthyl ring. The substitution on W includes replacing one or more —H with —OH, alkyl, O-alkyl, branched alkyl, or cycloalkyl, containing 1-6 carbon atoms or combinations thereof. Y is a substituted or unsubstituted phenyl ring or substituted or unsubstituted naphthyl ring. The substitution for Y includes replacement of one or more —H atoms with CN, CF3, NO2, methoxy, benzoyl, phenoxy, phenoxymethyl or combinations thereof. These compounds are useful as antibacterial against gram negative and gram positive bacteria and as antiinflammatory agents.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.