O-alkylated rapamycin derivatives and their use, particularly as immunosuppressants
US6440990B1 · kind B1 · utility
49Cited by
9References
35Claims
0Family size
Assignee
Inventors
Key dates
| Filing date | May 23, 1997 |
| Grant date | Aug 27, 2002 |
| Priority date | — |
| Expiry date | May 23, 2017 |
Classification
- Technology area (CPC A)Human Necessities
- CPC primaryA61P43/00
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
Novel derivatives of rapamycin, particularly 9-deoxo-rapamycins, 26-dihydro-rapamycins, and 40-O-substituted and 28,40-O,O-disubstituted rapamycins. are found to have pharmaceutical utility, particularly as immunosuppressants.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.