Patent · US Expired

Method of producing submicron particles of a labile agent and use thereof

US6444223B1 · kind B1 · utility

4Cited by
18References
108Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 28, 1999
Grant dateSep 3, 2002
Priority date
Expiry dateMay 28, 2019

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P5/02
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to a sustained release composition comprising micron particles of labile agent and a method of preparing and using the sustained release composition. The invention further relates to micron particles of a labile agent and a method of preparing the micron particles. The method of the invention for preparing a composition for the sustained release of a labile agent, comprises forming a suspension comprising the labile agent dispersed in a polymer solution comprising at least one biocompatible polymer and at least one polymer solvent. The suspension is then wet milled to achieve micron particles of the labile agent. The polymer solvent is then removed resulting in a solid polymer/labile agent matrix. The method for preparing micron particles of a labile agent comprises forming a suspension comprising the labile agent, dispersed in a polymer solution comprising at least one biocompatible polymer and at least one polymer solvent, and wet milling of the suspension.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.