Patent · US Expired

Process for production of piperidine derivatives

US6448406B1 · kind B1 · utility

5Cited by
26References
70Claims
0Family size

Assignee

Inventors

Key dates

Filing dateAug 9, 2000
Grant dateSep 10, 2002
Priority date
Expiry dateAug 9, 2020

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D261/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention relates to a method for preparing piperidine derivative compounds by converting, with a piperidine compound, regioisomers having the formula: where Z is —CG1G2G3; G1, G2, and G3 are the same or different and are selected from the group consisting of OR8, SR8, and NR8R9; X3 is halogen, OR15, SR15, NR15R16, OSO2R15, or NHSO2R15; R8, R9, R15, and R16 are the same or different and are selected from the group consisting of hydrogen, an alkyl moiety, and an aryl moiety; and A is a substituent of its ring and is selected from the group consisting of hydrogen, halogens, alkyl, hydroxy, alkoxy, and other substituents.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.