Patent · US Expired

Process for the preparation of chemical compounds

US6469172B2 · kind B2 · utility

2Cited by
1References
9Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 5, 2001
Grant dateOct 22, 2002
Priority date
Expiry dateMar 5, 2021

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02P20/55
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

An improved and efficient synthesis for the preparation of 2-amino-6-[(4-aminopiperidin-1-yl]methyl]pyridine, an intermediate compound in the preparation of muscarinic M3 receptor antagonists, includes as a final step the removal of trimethylacetyl and an amino protecting group from 2-trimethylacetyl-amino-6-[(4-protected aminopiperidin-1-yl)methyl]pyridine.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.