Patent · US Expired

Biodegradable targetable microparticle delivery system

US6471996B1 · kind B1 · utility

81Cited by
8References
14Claims
0Family size

Assignee

Inventors

Key dates

Filing dateFeb 11, 2000
Grant dateOct 29, 2002
Priority date
Expiry dateFeb 11, 2020

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY10T428/2982
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Copolymers designed for use as particulate carriers containing functionalizable amino acid subunits for coupling with targeting ligand are described. The copolymers are polyesters composed of &agr;-hydroxy acid subunits such as D,L-lactide and &agr;-amino acid subunits such as serine or in the preferred embodiment, terpolymers of D,L-lactide and glycolide and &agr;-amino acid subunits such as serine. Stable vaccine preparations useful as delayed release formulations containing antigen(s) or antigen(s) and co-adjuvants encapsulated within or physically mixed with polymeric microparticles are described. The particulate carriers are useful for delivering agents to the immune system of a subject by mucosal or parenteral routes to produce immune responses, including antibody responses.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.