Patent · US Expired

Indole and 2,3-dihydroindole derivatives, their preparation and use

US6476035B1 · kind B1 · utility

4Cited by
2References
16Claims
0Family size

Inventors

Key dates

Filing dateJan 25, 2000
Grant dateNov 5, 2002
Priority date
Expiry dateJan 25, 2020

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D409/12
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention relates to indole and 2,3-dihydroindole derivatives having formula (I) or any of its any of its enantiometers or any mixture thereof, or an acid addition salt thereof, wherein A, R1, R2, R3, W, X, Y and Z are as described in the description. The compounds are potent serotonin reuptake inhibitors and have 5-HT1A receptor antagonistic activity.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.