Patent · US Expired

Formulations and methods for treatment of mucosal associated conditions with an immune response modifier

US6486168B1 · kind B1 · utility

193Cited by
33References
16Claims
0Family size

Assignee

Inventors

Key dates

Filing dateSep 29, 2000
Grant dateNov 26, 2002
Priority date
Expiry dateSep 29, 2020

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D471/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Immune response modifier (IRM) compounds—imidazoquinoline amines, imidazopyridine amines, 6,7-fused cycloalkylimidazopyridine amines, 1,2-bridged imidazoquinoline amines, thiazolo- and oxazolo-quinolinamines and pyridinamines, imidazonaphthyridine and tetrahydroimidazonaphthyridine amines—are useful for the treatment of conditions at and below the mucosal surfaces by administering a therapeutically effective amount of such compounds to the mucosal surface. Novel pharmaceutical formulations are provided. In one embodiment, the pharmaceutical formulations are advantageous for treatment of cervical conditions such as cervical dysplasias including cervical intraepithelial neoplasias.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.