Patent · US Expired

Preparation of camptothecin and of its derivatives

US6486320B2 · kind B2 · utility

0Cited by
4References
45Claims
0Family size

Assignee

Inventors

Key dates

Filing dateSep 14, 2001
Grant dateNov 26, 2002
Priority date
Expiry dateSep 14, 2021

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D471/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention relates to a novel process for preparation of camptothecin and of its derivatives by convergent synthesis starting from a 3-(aminomethyl)quinoline derivative and 5-hydroxy-5-ethyl-6-oxo-5,6-dihydropyrancarboxylic acid and to the intermediates obtained.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.