Patent · US Expired

Intrinsic dissolution apparatus with stationary sample holder

US6497157B1 · kind B1 · utility

12Cited by
13References
8Claims
0Family size

Assignee

Inventors

Key dates

Filing dateNov 13, 2000
Grant dateDec 24, 2002
Priority date
Expiry dateApr 2, 2021

Classification

  • Technology area (CPC G)Physics
  • CPC primaryG01N2013/006
  • WIPO fieldMeasurement
  • WIPO sectorInstruments

Abstract

For intrinsic dissolution testing, a drug pellet (i.e., the dissolution test sample) is retained within a cylindrical recess in a sample holder that is placed at the bottom of a dissolution vessel containing an appropriate dissolution medium with the sample holder oriented with the drug pellet facing up. During the testing cycle, the dissolution medium may be stirred, e.g., using a conventional USP 2 rotating paddle, while the sample holder (and drug pellet) remain stationary at the bottom of the vessel. The orientation of the drug pellet during testing (i.e., facing up) decreases the likelihood of retention of air bubbles formed at the surface of the drug pellet (which bubbles could otherwise decrease the effective dissolution rate), thereby providing more accurate and consistent intrinsic dissolution test results.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.