Patent · US Expired

Injectable pharmaceutical composition comprising coated particles of camptothecin

US6509027B2 · kind B2 · utility

4Cited by
39References
38Claims
0Family size

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Key dates

Filing dateFeb 12, 2001
Grant dateJan 21, 2003
Priority date
Expiry dateFeb 12, 2021

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K31/4745
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A pharmaceutical composition is provided which comprises an aqueous suspension of solid particles, the solid particles comprising a camptothecin, the solid particles having mean diameters between about 0.05 um and 10 um, the particles coated with a 0.3 nm to 3.0 um thick layer of a membrane-forming amphipathic lipid. The pharmaceutical composition is particularly well suited for delivering camptothecins, particularly 9-nitro-camptothecin intravenously.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.