Patent · US Expired

Method for administering camptothecins via injection of pharmaceutical composition comprising coated particles of a camptothecin

US6534080B2 · kind B2 · utility

5Cited by
6References
42Claims
0Family size

Assignees

Inventors

Key dates

Filing dateFeb 12, 2001
Grant dateMar 18, 2003
Priority date
Expiry dateFeb 12, 2021

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K31/4745
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A method for administering a camptothecin to a patient comprising: injecting into a patient a pharmaceutical composition comprising an aqueous suspension of solid particles suitable for intravenous delivery, the solid particles comprising a camptothecin, and a 0.3 nm to 3.0 &mgr;m thick layer of a membrane-forming amphipathic lipid wherein the solid particles have mean diameters between about 0.05 &mgr;m and 10 &mgr;m. The method is particularly well suited for delivering camptothecins, particularly 9-nitro-camptothecin intravenously.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.