Patent · US Expired

Substituted (aminoiminomethyl or aminomethyl) benzoheteroaryl compounds

US6541505B1 · kind B1 · utility

2Cited by
0References
35Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 30, 2000
Grant dateApr 1, 2003
Priority date
Expiry dateJun 30, 2020

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D491/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

This invention is directed to an (aminoiminomethyl or aminomethyl)benzoheteroaryl compound of formula I which is useful for inhibiting the activity of Factor Xa by combining said compound with a composition containing Factor Xa. The present invention is also directed to compositions containing compounds of the formula I, methods for their preparation, their use, such as in inhibiting the formation of thrombin or for treating a patient suffering from, or subject to, a disease state associated with a physiologically detrimental excess amount of thrombin.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.