Patent · US Expired

Methods of synthesizing sultams and anti-viral compositions

US6562850B1 · kind B1 · utility

1Cited by
1References
8Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 15, 1999
Grant dateMay 13, 2003
Priority date
Expiry dateJul 15, 2019

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D275/06
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The invention relates to a new class of compounds herein identified generally as “sultams”, which may be represented by the following formula V, in FIG. 1, in which numbering of the atoms is started with the sulfur atom of the isothiazole. Two of the rings (rings A and C) are aromatic, and the third is a heterocyclic ring (ring B), a cyclic sulfonamide. Of particular importance are the enantiomerically pure sultams since they are especially potent HIV-1 inhibitors.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.