Patent · US Expired

Lactonization process

US6562984B2 · kind B2 · utility

4Cited by
10References
20Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 11, 2002
Grant dateMay 13, 2003
Priority date
Expiry dateMar 11, 2022

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P3/06
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Lactonization of statins can be achieved using a lactonization agent that forms a hydrated complex with the produced water that is insoluble in the reaction solvent. By binding the produced water in an insoluble complex, the reaction is pulled to the lactone side, using mild conditions in short reactions times and with reduced risk of impurities.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.