Preparation of anhydrous CETP inhibitor
US6573383B2 · kind B2 · utility
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14Claims
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Assignee
Inventor
Key dates
| Filing date | Sep 27, 2002 |
| Grant date | Jun 3, 2003 |
| Priority date | — |
| Expiry date | Sep 27, 2022 |
Classification
- Technology area (CPC A)Human Necessities
- CPC primaryA61P25/02
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
This invention relates to methods for preparing anhydrous CETP inhibitor, (2R,4S)-4-[(3,5-bis-trifluoromethyl-benzyl)-methoxycarbonyl-amino]-2-ethyl-6-trifluoromethyl-3,4-dihydro-2H-quinoline-1-carboxylic acid ethyl ester.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.