Patent · US Expired

Method of ameliorating erectile dysfunction

US6586391B1 · kind B1 · utility

2Cited by
5References
12Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 18, 2000
Grant dateJul 1, 2003
Priority date
Expiry dateJul 18, 2020

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P43/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The mechanism of hypertension following acute NO synthase blockage is via endothelin-mediated vasoconstriction. Thus, NO appears to inhibit endothelin activity by blocking its expression and not as a chronic direct acting vasodilator. Administration of an endothelin antagonist to a patient in a ‘normal’ physiological state may result in specific regional vasodilation. This treatment finds utility in the treatment of erectile dysfunction.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.